Skip to content

Florida shipping only this week. All states soon. Sign up for updates →

Retatrutide compounded injection vial

// Weight Loss

Retatrutide

Triple agonist (GLP-1 + GIP + glucagon). Newer mechanism, strong early data.

  • Triple-pathway agonist · GLP-1 + GIP + glucagon
  • Highest reported weight-loss signal of compounded GLP-class options
  • Compounded under USP 797 sterile standards
  • Three vial sizes for titration and maintenance

Starting from

Sign-in required. A licensed physician reviews every prescription before it ships.

Read the full protocol ↓

// All formulations

3 formulations available

For orientation only — your physician confirms the final protocol on the pharmacy storefront.

OptionSizePrice
Introductory · 1 mL1 mL vial$263
Standard · 3 mL3 mL vial$371
Best value · 5 mL5 mL vial$433

Compounded by Greenstone Rx · Florida 503A pharmacy

Continue to Pharmacy →

// The science

About Retatrutide

Retatrutide is a triple agonist — activating GLP-1, GIP, and glucagon receptors simultaneously. In Phase 2 trials, retatrutide produced the largest average weight-loss signals to date. Compounded as an injectable at 20 mg/mL across three vial sizes for stepped titration.

// How it works

How it works

Retatrutide activates three receptors: GLP-1, GIP, and glucagon. The glucagon arm increases energy expenditure — your body burns more calories at rest — which differentiates it from the dual agonists.

// Who it's for

Who it's for

Patients who haven't reached their goal on tirzepatide or semaglutide. Those whose providers think additional metabolic-rate effect would help. Phase 2 trial data show some patients losing 24%+ at the highest doses.

// What to expect

Your timeline

Slow ramp over 4–8 months. Higher peak doses than other GLP-1s. Side-effect profile similar to tirzepatide; nausea on dose increases.

// Who should not take this

Who should not take this

Same family of contraindications as semaglutide and tirzepatide. As a newer molecule, screening is even more careful.

// Typical starting dose

Typical starting dose

A typical starting protocol is 2 mg once weekly, with slow titration over 4–8 months toward a higher peak dose than other GLP-1s. Suggestions only — your physician reviews and approves the final protocol before any medication ships.

// Ready when you are

Start your prescription.

You'll complete a short health screening on the pharmacy storefront. A licensed physician reviews every order before any medication ships.

Continue to Pharmacy →

Compounded by a 503A licensed pharmacy pursuant to a valid prescription. Not an FDA-approved drug. Not intended to diagnose, treat, cure, or prevent any disease. Individual results vary. Full disclaimer.